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Tertiapin Q, CAS 252198-49-5

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  • Tertiapin Q, blocker of inward-rectifier r K+ channels

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Description

  • Product name

    Tertiapin Q, blocker of inward-rectifier r K+ channels

  • Description

    Potent inward rectifier K+ channel blocker

  • Biological description

    Potent blocker of inward rectifier K+ channels. Stable analog of the bee venom tertiapin. High affinity for ROMK1 and GIRK1/4 (Ki values are 1.3 and 13.3 nM, respectively).

  • Purity

    > 95%

  • CAS Number

    252198-49-5
  • Molecular Formula: C106H175N35O24S4

  • Chemical structure

    Tertiapin-Q [252198-49-5]

  • References

    1. Drici, M.D. et al. (2000) Br. J. Pharmacol. 131, 569.

    2. mura, H. et al. (2000) J. Pharmacol. Exp. Ther. 293, 196.

    3. Peleg, S. et al. (2002) Neuron 33, 87.